Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Arginase (Leishmania amazonensis) | BDBM50241867 (((2R,3R,4R,5R,6R)-6-(3,4-dihydroxyphenethoxy)-5-hy...) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Similars | Article PubMed | 700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal de S£o Carlos Curated by ChEMBL | Assay Description Competitive inhibition of Leishmania amazonensis arginase assessed as inhibition constant for enzyme-inhibitor complex using L-arginine as substrate ... | J Nat Prod 79: 1459-63 (2016) Article DOI: 10.1021/acs.jnatprod.5b00875 BindingDB Entry DOI: 10.7270/Q2G73J78 | |||||||||||
More data for this Ligand-Target Pair |