Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Aromatase (Homo sapiens (Human)) | BDBM50049763![]() (2-[1-(3H-Imidazol-4-yl)-meth-(E)-ylidene]-3,4-dihy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a | n/a |
Universität de Saarlandes Curated by ChEMBL | Assay Description In vitro inhibitory activity against Cytochrome P450 19A1 using human placental microsomes. | J Med Chem 39: 834-41 (1996) Article DOI: 10.1021/jm950377t BindingDB Entry DOI: 10.7270/Q29K499J | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Rattus norvegicus) | BDBM50049763![]() (2-[1-(3H-Imidazol-4-yl)-meth-(E)-ylidene]-3,4-dihy...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 170 | n/a | n/a | n/a | n/a | n/a | n/a |
American University of Ras Al Khaimah Curated by ChEMBL | Assay Description Inhibition of rat ovarian aromatase | Eur J Med Chem 102: 375-86 (2015) Article DOI: 10.1016/j.ejmech.2015.08.010 BindingDB Entry DOI: 10.7270/Q2ZC84Q6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Aromatase (Homo sapiens (Human)) | BDBM50049763![]() (2-[1-(3H-Imidazol-4-yl)-meth-(E)-ylidene]-3,4-dihy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 260 | n/a | n/a | n/a | n/a | n/a | n/a |
Universität de Saarlandes Curated by ChEMBL | Assay Description In vitro inhibitory activity against Cytochrome P450 19A1 using human placental microsomes. | J Med Chem 39: 834-41 (1996) Article DOI: 10.1021/jm950377t BindingDB Entry DOI: 10.7270/Q29K499J | |||||||||||
More data for this Ligand-Target Pair |