Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Beta-1 adrenergic receptor (GUINEA PIG) | BDBM50404791![]() (CHEMBL31025) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | 316 | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation | J Med Chem 25: 1408-12 (1983) BindingDB Entry DOI: 10.7270/Q2S183PB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (GUINEA PIG) | BDBM50404791![]() (CHEMBL31025) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | 0.00000100 | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 3h | J Med Chem 25: 1408-12 (1983) BindingDB Entry DOI: 10.7270/Q2S183PB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Beta-1 adrenergic receptor (GUINEA PIG) | BDBM50404791![]() (CHEMBL31025) | PDB UniProtKB/TrEMBL GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | n/a | 100 | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Ability to block Beta-1 adrenergic receptor in guinea pig right atria preparation at a duration of 40 min | J Med Chem 25: 1408-12 (1983) BindingDB Entry DOI: 10.7270/Q2S183PB | |||||||||||
More data for this Ligand-Target Pair |