Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Bromodomain adjacent to zinc finger domain protein 2B (Homo sapiens (Human)) | BDBM50277366 (CHEMBL4171398) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | n/a | 5.40E+4 | n/a | n/a | n/a | n/a | n/a |
University of Z£rich Curated by ChEMBL | Assay Description Binding affinity to human BAZ2B (S2054 to S2168 residues) expressed in bacterial expression system by BROMOscan assay | Eur J Med Chem 139: 564-572 (2017) Article DOI: 10.1016/j.ejmech.2017.08.028 BindingDB Entry DOI: 10.7270/Q2833VJS | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) |