BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 4' and Ligand = 'BDBM329752'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Bromodomain-containing protein 4


(Homo sapiens (Human))		BDBM329752
PNG
(Preparation of 2-[6-(4-chlorophenyl)-1-methyl-4H-[...)
Show SMILES Cc1nnc2C(CC(=O)N3CC(F)C3)C=C(c3ccc(Cl)cc3)c3ccccc3-n12 |t:15|
Show InChI InChI=1S/C23H20ClFN4O/c1-14-26-27-23-16(11-22(30)28-12-18(25)13-28)10-20(15-6-8-17(24)9-7-15)19-4-2-3-5-21(19)29(14)23/h2-10,16,18H,11-13H2,1H3
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 220n/an/an/an/an/an/a



BAYER PHARMA AKTIENGESELLSCHAFT

US Patent


Assay Description
For this purpose, a time-resolved fluorescence resonance energy transfer (TR-FRET) assay was used, which measures the binding between N-terminally Hi...

US Patent US9663523 (2017)


BindingDB Entry DOI: 10.7270/Q2NC639V
More data for this
Ligand-Target Pair