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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 9 [134-239]' and Ligand = 'BDBM321409'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Bromodomain-containing protein 9 [134-239]


(Homo sapiens (Human))		BDBM321409
PNG
(6-[(E)-but-2-enyl]-4-[3-chloro-4-(pyrrolidine-1-ca...)
Show SMILES C\C=C\Cn1cc(-c2ccc(C(=O)N3CCCC3)c(Cl)c2)c2cc(C)[nH]c2c1=O
Show InChI InChI=1S/C23H24ClN3O2/c1-3-4-9-27-14-19(18-12-15(2)25-21(18)23(27)29)16-7-8-17(20(24)13-16)22(28)26-10-5-6-11-26/h3-4,7-8,12-14,25H,5-6,9-11H2,1-2H3/b4-3+
PDB

UniProtKB/SwissProt

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PC cid
PC sid
UniChem
US Patent
n/an/a 10n/an/an/an/an/an/a



GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent


Assay Description
His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...

US Patent US10183009 (2019)


BindingDB Entry DOI: 10.7270/Q2125VRQ
More data for this
Ligand-Target Pair