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Found 1 hit Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 9 [134-239]' and Ligand = 'BDBM321417'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Bromodomain-containing protein 9 [134-239]


(Homo sapiens (Human))		BDBM321417
PNG
(6-allyl-4-[3-chloro-4-(morpholine-4-carbonyl)pheny...)
Show SMILES Cc1cc2c(cn(CC=C)c(=O)c2[nH]1)-c1ccc(C(=O)N2CCOCC2)c(Cl)c1
Show InChI InChI=1S/C22H22ClN3O3/c1-3-6-26-13-18(17-11-14(2)24-20(17)22(26)28)15-4-5-16(19(23)12-15)21(27)25-7-9-29-10-8-25/h3-5,11-13,24H,1,6-10H2,2H3
PDB

UniProtKB/SwissProt

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PC cid
PC sid
UniChem
US Patent
n/an/a 12n/an/an/an/an/an/a



GENENTECH, INC.; CONSTELLATION PHARMACEUTICALS, INC.

US Patent


Assay Description
His/Flag epitope tagged BRD9134-239 was cloned, expressed, and purified to homogeneity. BRD9 binding and inhibition was assessed by monitoring the en...

US Patent US10183009 (2019)


BindingDB Entry DOI: 10.7270/Q2125VRQ
More data for this
Ligand-Target Pair