Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'CREB-binding protein [1081-1197]' and Ligand = 'BDBM511385'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
CREB-binding protein [1081-1197] (Homo sapiens (Human))	BDBM511385 (N-methyl-1-(3-(1-methyl- 1H-pyrazol-3- yl)isoquino...) Show SMILES CNC(=O)N1CCn2c(C1)c(nc2C1CCOCC1)-c1cccc2cc(ncc12)-c1cnn(C)c1 Show InChI	PDB MMDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2	n/a	n/a	n/a	n/a	n/a	n/a
TBA					Assay Description 5 nM GST-CBP(1081-1197) and 20 nM biotin-H4(1-21) Ac-K5/8/12/16 (AnaSpec. 64989) were incubated with varying concentrations of CBP inhibitors in 15 &...				Citation and Details BindingDB Entry DOI: 10.7270/Q2CC13VN
					More data for this Ligand-Target Pair