Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cannabinoid receptor 1 (Homo sapiens (Human)) | BDBM50562158![]() (CHEMBL4747585) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University Curated by ChEMBL | Assay Description Displacement of [3H]CP55940 from human CB1 receptor incubated for 90 mins by radioligand binding assay | Bioorg Med Chem Lett 13: 1119-23 (2003) Article DOI: 10.1016/j.ejmech.2020.112857 BindingDB Entry DOI: 10.7270/Q2D21X0K | |||||||||||
More data for this Ligand-Target Pair |