Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Carboxypeptidase A1 (Homo sapiens (Human)) | BDBM50373038 (CHEMBL407567) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL DrugBank MMDB PC cid PC sid PDB UniChem Similars | DrugBank Article PubMed | 150 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Yanbian University Curated by ChEMBL | Assay Description Inhibition of CPA | Bioorg Med Chem 16: 3596-601 (2008) Article DOI: 10.1016/j.bmc.2008.02.010 BindingDB Entry DOI: 10.7270/Q25Q4WZ7 | |||||||||||
More data for this Ligand-Target Pair |