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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Casein kinase 1, delta tv1' and Ligand = 'BDBM50488798'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Casein kinase 1, delta tv1


(Sus scrofa)		BDBM50488798
PNG
(CHEMBL2295944)
Show SMILES CCC[C@H](O)Nc1nc(Nc2cccc(c2)-c2cncnc2)c2ncn(C(C)C)c2n1 |r|
Show InChI InChI=1S/C22H26N8O/c1-4-6-18(31)27-22-28-20(19-21(29-22)30(13-25-19)14(2)3)26-17-8-5-7-15(9-17)16-10-23-12-24-11-16/h5,7-14,18,31H,4,6H2,1-3H3,(H2,26,27,28,29)/t18-/m0/s1
PDB

UniProtKB/TrEMBL

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
Article
n/an/a 200n/an/an/an/an/an/a


TBA

Assay Description
Inhibition of Sus scrofa (pig) casein kinase 1delta/epsilon isolated from brain using RRKHAAIGpSAYSITA and [gamma33P]ATP as substrate after 30 min by...

Citation and Details

Article DOI: 10.1007/s00044-012-0334-1
BindingDB Entry DOI: 10.7270/Q2ZP490F
More data for this
Ligand-Target Pair