Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cholecystokinin receptor type A (RAT) | BDBM50003666![]() (3-[2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 0.0500 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against cholecystokinin type A receptor from rat pancreas binding assay | J Med Chem 35: 4249-52 (1992) BindingDB Entry DOI: 10.7270/Q2Z60N07 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cholecystokinin receptor type A (Homo sapiens (Human)) | BDBM50003666![]() (3-[2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Roche Research Center Curated by ChEMBL | Assay Description Inhibitory activity against cholecystokinin type A receptor from bovine striatal binding assay | J Med Chem 35: 4249-52 (1992) BindingDB Entry DOI: 10.7270/Q2Z60N07 | |||||||||||
More data for this Ligand-Target Pair |