Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Chromodomain Y-like protein (Homo sapiens (Human)) | BDBM50194259 (CHEMBL3939958) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 910 | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Binding affinity to human N-terminal GST-tagged CDYL1b chromodomain (1 to 78 residues) expressed in Escherichia coli Rosetta BL21(DE3)pLysS by ITC me... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromodomain Y-like protein (Homo sapiens (Human)) | BDBM50194259 (CHEMBL3939958) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 910 | n/a | n/a | n/a | n/a | n/a |
Peking University Curated by ChEMBL | Assay Description Binding affinity to CDYL chromodomain (unknown origin) by isothermal titration calorimetry | Eur J Med Chem 182: (2019) Article DOI: 10.1016/j.ejmech.2019.111656 BindingDB Entry DOI: 10.7270/Q23N26R6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromodomain Y-like protein (Homo sapiens (Human)) | BDBM50194259 (CHEMBL3939958) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 5.60E+3 | n/a | n/a | n/a | n/a | n/a |
Peking University Curated by ChEMBL | Assay Description Binding affinity to recombinant human N-terminal GST-tagged CDYL (1 to 60 residues) expressed in Escherichia coli BL2 by SPR analysis | Eur J Med Chem 182: (2019) Article DOI: 10.1016/j.ejmech.2019.111656 BindingDB Entry DOI: 10.7270/Q23N26R6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromodomain Y-like protein (Homo sapiens (Human)) | BDBM50194259 (CHEMBL3939958) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | 910 | n/a | n/a | n/a | n/a | n/a |
University of Connecticut Curated by ChEMBL | Assay Description Binding affinity to CDYL1b (unknown origin) after 30 mins by fluorescence polarization assay | Eur J Med Chem 136: 14-35 (2017) Article DOI: 10.1016/j.ejmech.2017.04.047 BindingDB Entry DOI: 10.7270/Q2F76G3G | |||||||||||
More data for this Ligand-Target Pair |