Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cyclin-K/Cyclin-dependent kinase 12 (Homo sapiens (Human)) | BDBM572066![]() ((R)-N-(4-(3-(pyrido[3,4-d]pyrimidin- 2-ylamino)pyr...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | US Patent | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description A radiometric protein kinase assay (33PanQinaseŽ Activity Assay) was used for measuring the kinase activity of the three protein kinases. All kinase ... | Citation and Details BindingDB Entry DOI: 10.7270/Q2CF9TBB | |||||||||||
More data for this Ligand-Target Pair |