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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Cystic fibrosis transmembrane conductance regulator [1-507,509-1480]' and Ligand = 'BDBM526470'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Cystic fibrosis transmembrane conductance regulator [1-507,509-1480]


(Homo sapiens (Human))		BDBM526470
PNG
(US11186566, Compound 9)
Show SMILES CC1(C)CC(CO)CN1c1nc(ccc1C(=O)NS(=O)(=O)c1ccccc1)-n1ccc(OCCC2(CC2)C(F)(F)F)n1
PDB

UniProtKB/SwissProt

GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/an/an/a 550n/an/an/an/a


TBA

Assay Description
The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...

Citation and Details

BindingDB Entry DOI: 10.7270/Q22R3VVH
More data for this
Ligand-Target Pair