Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
D(1A) dopamine receptor (RAT) | BDBM50300159 (CHEMBL583422 | Ethyl 5-(3-(4-((benzo[d][1,3]dioxol...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ di Napoli Curated by ChEMBL | Assay Description Displacement of [3H]SCH23390 from dopamine D1 in rat striatum by liquid scintillation counting | Eur J Med Chem 45: 752-9 (2010) Article DOI: 10.1016/j.ejmech.2009.11.023 BindingDB Entry DOI: 10.7270/Q2445MJR | |||||||||||
More data for this Ligand-Target Pair |