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Found 1 hit Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM50000573'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
D(2) dopamine receptor


(Rattus norvegicus (rat))		BDBM50000573
PNG
(6-{6-[2-(2-Hydroxy-ethyl)-piperidin-4-yl]-hexyloxy...)
Show SMILES OCCC1CC(CCCCCCOc2ccc3oc(cc(=O)c3c2)-c2ccccc2)CCN1
Show InChI InChI=1S/C28H35NO4/c30-16-14-23-18-21(13-15-29-23)8-4-1-2-7-17-32-24-11-12-27-25(19-24)26(31)20-28(33-27)22-9-5-3-6-10-22/h3,5-6,9-12,19-21,23,29-30H,1-2,4,7-8,13-18H2
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PC sid
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Similars
PubMed
 2.70E+3n/an/an/an/an/an/an/an/a



Nova Pharmaceutical Corporation

Curated by ChEMBL


Assay Description
Affinity towards dopamine receptor D2 was determined by competition studies using [3H]-sulpiride in rat striatum.

J Med Chem 35: 1526-35 (1992)


BindingDB Entry DOI: 10.7270/Q2XG9Q38
More data for this
Ligand-Target Pair