Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Endoplasmic reticulum aminopeptidase 2 (Homo sapiens (Human)) | BDBM50245396 (CHEMBL4101200) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 37 | n/a | n/a | n/a | n/a | n/a | n/a |
National and Kapodistrian University of Athens Curated by ChEMBL | Assay Description Inhibition of ERAP2 (unknown origin) expressed in Hi5 cells by in vitro fluorimetric assay | J Med Chem 59: 9107-9123 (2016) Article DOI: 10.1021/acs.jmedchem.6b01031 BindingDB Entry DOI: 10.7270/Q2PK0JJG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endoplasmic reticulum aminopeptidase 2 (Homo sapiens (Human)) | BDBM50245396 (CHEMBL4101200) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 37 | n/a | n/a | n/a | n/a | n/a | n/a |
Wroc?aw University of Science and Technology Curated by ChEMBL | Assay Description Inhibition of ERAP2 (unknown origin) | Bioorg Med Chem Lett 29: 1031-1042 (2019) Article DOI: 10.1016/j.bmcl.2019.02.034 BindingDB Entry DOI: 10.7270/Q2DR2ZSK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endoplasmic reticulum aminopeptidase 2 (Homo sapiens (Human)) | BDBM50245396 (CHEMBL4101200) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of human ERAP2 | Citation and Details Article DOI: 10.1016/j.ejmech.2020.113053 BindingDB Entry DOI: 10.7270/Q29Z98PR | |||||||||||
More data for this Ligand-Target Pair |