Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50289937 (3-(4-Chloro-3-methyl-isoxazol-5-ylsulfamoyl)-thiop...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article | n/a | n/a | 148 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description In vitro binding affinity in a radioligand binding experiment by competition with [125I]-labeled endothelin-1 for ETA receptor | Bioorg Med Chem Lett 7: 2093-2098 (1997) Article DOI: 10.1016/S0960-894X(97)00367-3 BindingDB Entry DOI: 10.7270/Q2WH2PZF | |||||||||||
More data for this Ligand-Target Pair |