Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Excitatory amino acid transporter 1 (Homo sapiens (Human)) | BDBM50107948 (2-Amino-3-(2-hydroxy-2H-pyrazol-3-yl)-propionic ac...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
The Royal Danish School of Pharmacy Curated by ChEMBL | Assay Description Binding affinity for Excitatory amino acid transporter 1 (EAAT-1) in Glu uptake system | J Med Chem 45: 19-31 (2001) BindingDB Entry DOI: 10.7270/Q2KH0MMK | |||||||||||
More data for this Ligand-Target Pair |