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Found 1 hit Enz. Inhib. hit(s) with Target = 'Fatty-acid amide hydrolase 1' and Ligand = 'BDBM50236341'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Fatty-acid amide hydrolase 1


(Homo sapiens (Human))		BDBM50236341
PNG
(CHEMBL4102620)
Show SMILES COc1ccccc1N1CCN(CCCCNC(=O)Oc2ccc(c(OC)c2)-c2cccc(c2)C(N)=O)CC1
Show InChI InChI=1S/C30H36N4O5/c1-37-27-11-4-3-10-26(27)34-18-16-33(17-19-34)15-6-5-14-32-30(36)39-24-12-13-25(28(21-24)38-2)22-8-7-9-23(20-22)29(31)35/h3-4,7-13,20-21H,5-6,14-19H2,1-2H3,(H2,31,35)(H,32,36)
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n/an/a 63n/an/an/an/an/an/a



Universit£ di Bologna

Curated by ChEMBL


Assay Description
Inhibition of human FAAH1 expressed in HEK293 cell membrane-enriched lysate using AMC arachidonyl amide as substrate preincubated for 50 mins followe...

J Med Chem 60: 2287-2304 (2017)


Article DOI: 10.1021/acs.jmedchem.6b01578
BindingDB Entry DOI: 10.7270/Q29S1T9P
More data for this
Ligand-Target Pair