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Found 1 hit Enz. Inhib. hit(s) with Target = 'Fatty-acid amide hydrolase 1' and Ligand = 'BDBM50236349'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Fatty-acid amide hydrolase 1


(Homo sapiens (Human))		BDBM50236349
PNG
(CHEMBL4072140)
Show SMILES Clc1cccc(N2CCN(CCCCNC(=O)Oc3ccc4c(c3)[nH]c3ccccc43)CC2)c1Cl
Show InChI InChI=1S/C27H28Cl2N4O2/c28-22-7-5-9-25(26(22)29)33-16-14-32(15-17-33)13-4-3-12-30-27(34)35-19-10-11-21-20-6-1-2-8-23(20)31-24(21)18-19/h1-2,5-11,18,31H,3-4,12-17H2,(H,30,34)
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n/an/a 8n/an/an/an/an/an/a



Universit£ di Bologna

Curated by ChEMBL


Assay Description
Inhibition of human FAAH1 expressed in HEK293 cell membrane-enriched lysate using AMC arachidonyl amide as substrate preincubated for 50 mins followe...

J Med Chem 60: 2287-2304 (2017)


Article DOI: 10.1021/acs.jmedchem.6b01578
BindingDB Entry DOI: 10.7270/Q29S1T9P
More data for this
Ligand-Target Pair