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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Fibroblast growth factor receptor 4' and Ligand = 'BDBM50240573'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Fibroblast growth factor receptor 4


(Homo sapiens (Human))		BDBM50240573
PNG
(CHEMBL4077859)
Show SMILES COc1cc(OC)c(F)c(COc2cnc(N[C@@H]3COC[C@@H]3NC(=O)C=C)nc2)c1F |r|
Show InChI InChI=1S/C20H22F2N4O5/c1-4-17(27)25-13-9-30-10-14(13)26-20-23-6-11(7-24-20)31-8-12-18(21)15(28-2)5-16(29-3)19(12)22/h4-7,13-14H,1,8-10H2,2-3H3,(H,25,27)(H,23,24,26)/t13-,14+/m0/s1
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Article
PubMed
n/an/a 13n/an/an/an/an/an/a



WuXi AppTec (Shanghai) Co., Ltd.

Curated by ChEMBL


Assay Description
Inhibition of recombinant human N-terminal His-tagged FGFR4 cytoplasmic domain (781 to 133 residues) expressed in baculovirus expression system using...

Bioorg Med Chem Lett 27: 2420-2423 (2017)


Article DOI: 10.1016/j.bmcl.2017.04.014
BindingDB Entry DOI: 10.7270/Q2M90BT6
More data for this
Ligand-Target Pair