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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Free fatty acid receptor 1' and Ligand = 'BDBM50271611'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Free fatty acid receptor 1


(Homo sapiens (Human))		BDBM50271611
PNG
(CHEMBL4125720)
Show SMILES Clc1ccc2ccn(CCOc3ccc(CC4SC(=O)NC4=O)cc3)c2c1
Show InChI InChI=1S/C20H17ClN2O3S/c21-15-4-3-14-7-8-23(17(14)12-15)9-10-26-16-5-1-13(2-6-16)11-18-19(24)22-20(25)27-18/h1-8,12,18H,9-11H2,(H,22,24,25)
PDB

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PC cid
PC sid
UniChem

Similars
Article
PubMed
n/an/an/an/a 5.06E+3n/an/an/an/a



Suez Canal University

Curated by ChEMBL


Assay Description
Transactivation of recombinant human FFAR1 expressed in CHOK1 cells co-expressing Galpha15 assessed as increase in calcium flux measured after 20 sec...

Bioorg Med Chem Lett 28: 1595-1602 (2018)


Article DOI: 10.1016/j.bmcl.2018.03.051
BindingDB Entry DOI: 10.7270/Q2N58PVR
More data for this
Ligand-Target Pair