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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Free fatty acid receptor 1' and Ligand = 'BDBM50271615'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Free fatty acid receptor 1


(Homo sapiens (Human))		BDBM50271615
PNG
(CHEMBL4130213)
Show SMILES FC(F)(F)c1ccc(cc1)C(OCCOc1ccc(CC2SC(=O)NC2=O)cc1)c1ccccc1
Show InChI InChI=1S/C26H22F3NO4S/c27-26(28,29)20-10-8-19(9-11-20)23(18-4-2-1-3-5-18)34-15-14-33-21-12-6-17(7-13-21)16-22-24(31)30-25(32)35-22/h1-13,22-23H,14-16H2,(H,30,31,32)
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Similars
Article
PubMed
n/an/an/an/a 1.13E+4n/an/an/an/a



Suez Canal University

Curated by ChEMBL


Assay Description
Transactivation of recombinant human FFAR1 expressed in CHOK1 cells co-expressing Galpha15 assessed as increase in calcium flux measured after 20 sec...

Bioorg Med Chem Lett 28: 1595-1602 (2018)


Article DOI: 10.1016/j.bmcl.2018.03.051
BindingDB Entry DOI: 10.7270/Q2N58PVR
More data for this
Ligand-Target Pair