BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'G protein-activated inward rectifier potassium channel 1/4' and Ligand = 'BDBM585718'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
G protein-activated inward rectifier potassium channel 1/4


(Homo sapiens (Human))
BDBM585718
PNG
((S)-8-chloro-1-(2,6- dichlorophenyl)-5-((2,3- dihy...)
Show SMILES Cc1cc(=O)c2c(NC[C@H](O)CO)ncc(Cl)c2n1-c1c(Cl)cccc1Cl |r,wD:9.9,(4.67,-.14,;3.33,-.91,;3.33,-2.45,;2,-3.22,;2,-4.76,;.67,-2.45,;-.67,-3.22,;-.67,-4.76,;-2,-5.53,;-3.33,-4.76,;-4.67,-5.53,;-3.33,-3.22,;-4.67,-2.45,;-2,-2.45,;-2,-.91,;-.67,-.14,;-.67,1.4,;.67,-.91,;2,-.14,;2,2.45,;.67,3.22,;-.67,2.45,;.67,4.76,;2,5.53,;3.33,4.76,;3.33,3.22,;4.67,2.45,)|
PDB

UniProtKB/SwissProt

antibodypedia
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 15n/an/an/an/an/an/a


TBA

Assay Description
Quattro is controlled using IonWorks v2 software to perform the following steps:a. Add 3.5 ul cells plus 3.5 ul external buffer to wells of Quattro P...


Citation and Details

BindingDB Entry DOI: 10.7270/Q2K64NXF
More data for this
Ligand-Target Pair