Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'G protein-activated inward rectifier potassium channel 4' and Ligand = 'BDBM50532011'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
G protein-activated inward rectifier potassium channel 4 (Homo sapiens (Human))	BDBM50532011 (CHEMBL4541815) Show SMILES Cc1cc(NC(=O)Cn2nnc(n2)-c2cc(Cl)cc(Cl)c2)n(n1)C1CCCCC1 Show InChI InChI=1S/C19H21Cl2N7O/c1-12-7-17(28(24-12)16-5-3-2-4-6-16)22-18(29)11-27-25-19(23-26-27)13-8-14(20)10-15(21)9-13/h7-10,16H,2-6,11H2,1H3,(H,22,29)	Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	n/a	2.12E+3	n/a	n/a	n/a	n/a
University of Nebraska Medical Center Curated by ChEMBL					Assay Description Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assay				Bioorg Med Chem Lett 29: 791-796 (2019) Article DOI: 10.1016/j.bmcl.2019.01.027 BindingDB Entry DOI: 10.7270/Q2BV7M47
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