Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
G-protein coupled bile acid receptor 1 (Homo sapiens (Human)) | BDBM50540724![]() (CHEMBL4646264) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2.26E+3 | n/a | n/a | n/a | n/a |
University of Naples "Federico II" Curated by ChEMBL | Assay Description Agonist activity at human GPBAR1 receptor expressed in HEK293T cells after 18 hrs by cAMP response element driven renilla-luciferase dual reporter ge... | ACS Med Chem Lett 11: 818-824 (2020) Article DOI: 10.1021/acsmedchemlett.9b00636 BindingDB Entry DOI: 10.7270/Q2DV1PD0 | |||||||||||
More data for this Ligand-Target Pair |