Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Gamma-aminobutyric acid receptor subunit alpha-3 (Homo sapiens (Human)) | BDBM50034820 (8-Chloro-3-methoxymethyl-5-methyl-4,5-dihydro-2,5,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Moltech Corporation Curated by ChEMBL | Assay Description Binding affinity to GABAA alpha-3-beta-3-gamma-2 receptor | J Med Chem 51: 3788-803 (2008) Article DOI: 10.1021/jm701433b BindingDB Entry DOI: 10.7270/Q2FQ9XH6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gamma-aminobutyric acid receptor subunit alpha-3 (Homo sapiens (Human)) | BDBM50034820 (8-Chloro-3-methoxymethyl-5-methyl-4,5-dihydro-2,5,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 328 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Sussex Curated by ChEMBL | Assay Description Binding affinity to GABA-A alpha3 (unknown origin) | J Med Chem 63: 3425-3446 (2020) Article DOI: 10.1021/acs.jmedchem.9b01312 BindingDB Entry DOI: 10.7270/Q2VD72WN | |||||||||||
More data for this Ligand-Target Pair |