Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Gastric inhibitory polypeptide receptor (Mus musculus) | BDBM50566469 (CHEMBL4876736) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at mouse GIPR expressed in CHO-K1 cells assessed as inhibition of GIP-induced cAMP production | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02069 BindingDB Entry DOI: 10.7270/Q23J3HQT | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Gastric inhibitory polypeptide receptor (Homo sapiens (Human)) | BDBM50566469 (CHEMBL4876736) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Antagonist activity at human GIPR expressed in HEK293 cells assessed as inhibition of GIP-induced cAMP production | Citation and Details Article DOI: 10.1021/acs.jmedchem.0c02069 BindingDB Entry DOI: 10.7270/Q23J3HQT | |||||||||||
More data for this Ligand-Target Pair |