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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Glucagon receptor' and Ligand = 'BDBM50110053'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Glucagon receptor


(Homo sapiens (Human))		BDBM50110053
PNG
(3-Chloro-4-hydroxy-benzoic acid [1-[4-(5-tert-buty...)
Show SMILES CC(C)(C)c1nc(COc2ccc(\C=N\NC(=O)c3ccc(O)c(Cl)c3)c3ccccc23)no1
Show InChI InChI=1S/C25H23ClN4O4/c1-25(2,3)24-28-22(30-34-24)14-33-21-11-9-16(17-6-4-5-7-18(17)21)13-27-29-23(32)15-8-10-20(31)19(26)12-15/h4-13,31H,14H2,1-3H3,(H,29,32)/b27-13+
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PC cid
PC sid
UniChem

Patents
PubMed
n/an/a 160n/an/an/an/an/an/a



Pfizer Global Research and Development

Curated by ChEMBL


Assay Description
In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagon

Bioorg Med Chem Lett 12: 663-6 (2002)


BindingDB Entry DOI: 10.7270/Q2J67G77
More data for this
Ligand-Target Pair