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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Glucagon receptor' and Ligand = 'BDBM50110059'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Glucagon receptor


(Homo sapiens (Human))		BDBM50110059
PNG
(3-Chloro-4-hydroxy-N-{2-[4-(4-isopropyl-benzyloxy)...)
Show SMILES COc1cc(CCNC(=N)c2ccc(O)c(Cl)c2)cc(OC)c1OCc1ccc(cc1)C(C)C
Show InChI InChI=1S/C27H31ClN2O4/c1-17(2)20-7-5-18(6-8-20)16-34-26-24(32-3)13-19(14-25(26)33-4)11-12-30-27(29)21-9-10-23(31)22(28)15-21/h5-10,13-15,17,31H,11-12,16H2,1-4H3,(H2,29,30)
PDB
MMDB

UniProtKB/SwissProt

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CHEMBL
PC cid
PC sid
UniChem
PubMed
n/an/a 5.20E+3n/an/an/an/an/an/a



Pfizer Global Research and Development

Curated by ChEMBL


Assay Description
In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagon

Bioorg Med Chem Lett 12: 663-6 (2002)


BindingDB Entry DOI: 10.7270/Q2J67G77
More data for this
Ligand-Target Pair