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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Glucagon receptor' and Ligand = 'BDBM50110078'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Glucagon receptor


(Homo sapiens (Human))		BDBM50110078
PNG
(3-Chloro-4-hydroxy-benzoic acid [1-[4-(4-isopropyl...)
Show SMILES CC(C)c1ccc(COc2ccc(\C=N\NC(=O)c3ccc(O)c(Cl)c3)cc2)cc1
Show InChI InChI=1S/C24H23ClN2O3/c1-16(2)19-7-3-18(4-8-19)15-30-21-10-5-17(6-11-21)14-26-27-24(29)20-9-12-23(28)22(25)13-20/h3-14,16,28H,15H2,1-2H3,(H,27,29)/b26-14+
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PC cid
PC sid
UniChem

Similars
PubMed
n/an/a 1.50E+3n/an/an/an/an/an/a



Pfizer Global Research and Development

Curated by ChEMBL


Assay Description
In vitro inhibitory activity against human glucagon receptor using [127I]-labeled glucagon

Bioorg Med Chem Lett 12: 663-6 (2002)


BindingDB Entry DOI: 10.7270/Q2J67G77
More data for this
Ligand-Target Pair