Found 2 hits Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, NMDA 1' and Ligand = 'BDBM86494' Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Glutamate receptor ionotropic, NMDA 1
(RAT) | BDBM86494
(EAA-090 | Perzinfotel | WAY-126090)Show SMILES [#8][P;v5]([#8])(=O)[#6]-[#6]-[#7]-1-[#6]-[#6]-[#6]-[#7]-c2c-1c(=O)c2=O Show InChI InChI=1S/C9H13N2O5P/c12-8-6-7(9(8)13)11(3-1-2-10-6)4-5-17(14,15)16/h10H,1-5H2,(H2,14,15,16) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| Purchase
MCE PC cid PC sid UniChem
Patents
| Article PubMed
| 28 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 310: 563-70 (2004)
Article DOI: 10.1124/jpet.104.066092 BindingDB Entry DOI: 10.7270/Q2DJ5D6D |
More data for this Ligand-Target Pair | |
Glutamate receptor ionotropic, NMDA 1
(RAT) | BDBM86494
(EAA-090 | Perzinfotel | WAY-126090)Show SMILES [#8][P;v5]([#8])(=O)[#6]-[#6]-[#7]-1-[#6]-[#6]-[#6]-[#7]-c2c-1c(=O)c2=O Show InChI InChI=1S/C9H13N2O5P/c12-8-6-7(9(8)13)11(3-1-2-10-6)4-5-17(14,15)16/h10H,1-5H2,(H2,14,15,16) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| Purchase
MCE PC cid PC sid UniChem
Patents
| Article PubMed
| 7.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Wyeth Research
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 310: 563-70 (2004)
Article DOI: 10.1124/jpet.104.066092 BindingDB Entry DOI: 10.7270/Q2DJ5D6D |
More data for this Ligand-Target Pair | |