Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histone deacetylase (Homo sapiens (Human)) | BDBM50483616 (CHEMBL1760912) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.39E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Menarini Ricerche Pomezia Curated by ChEMBL | Assay Description Inhibition of HDAC in human HeLa cells by fluorescent activity assay | Bioorg Med Chem Lett 21: 2305-8 (2011) Article DOI: 10.1016/j.bmcl.2011.02.085 BindingDB Entry DOI: 10.7270/Q2VQ35HJ | |||||||||||
More data for this Ligand-Target Pair |