Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histone deacetylase (Homo sapiens (Human)) | BDBM50492407![]() (CHEMBL2403449) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 3.79E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Menarini Ricerche Curated by ChEMBL | Assay Description Inhibition of HDAC in human HeLa cells assessed as deacetylation of substrate by fluorescence plate reader analysis | Bioorg Med Chem Lett 23: 4091-5 (2013) Article DOI: 10.1016/j.bmcl.2013.05.053 BindingDB Entry DOI: 10.7270/Q22F7RCD | |||||||||||
More data for this Ligand-Target Pair |