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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Importin subunit alpha-1' and Ligand = 'BDBM75000'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Importin subunit alpha-1


(Homo sapiens (Human))		BDBM75000
PNG
(2-methoxyethyl-[5-methyl-2-(p-tolyl)pyrazolo[1,5-a...)
Show SMILES COCCNc1cc(C)nc2cc(nn12)-c1ccc(C)cc1
Show InChI InChI=1S/C17H20N4O/c1-12-4-6-14(7-5-12)15-11-17-19-13(2)10-16(21(17)20-15)18-8-9-22-3/h4-7,10-11,18H,8-9H2,1-3H3
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MMDB

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PC cid
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n/an/an/an/a 3.77E+3n/an/an/an/a



Broad Institute

Curated by PubChem BioAssay


Assay Description
Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...

PubChem Bioassay (2010)


BindingDB Entry DOI: 10.7270/Q280513R
More data for this
Ligand-Target Pair