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Found 1 hit Enz. Inhib. hit(s) with Target = 'Lysine-specific demethylase 4C' and Ligand = 'BDBM263986'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Lysine-specific demethylase 4C


(Homo sapiens (Human))		BDBM263986
PNG
(2-{5-[(1-methyl-1H-indazol-6- yl)methoxy]-1H-pyraz...)
Show SMILES Cn1cc2ccc(COc3ccnn3-c3cc(ccn3)C(O)=O)cc2n1
Show InChI InChI=1S/C18H15N5O3/c1-22-10-14-3-2-12(8-15(14)21-22)11-26-17-5-7-20-23(17)16-9-13(18(24)25)4-6-19-16/h2-10H,11H2,1H3,(H,24,25)
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem
US Patent
n/an/a 550n/an/an/an/an/an/a



The Scripps Research Institute



Assay Description
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...

J Med Chem 50: 3359-68 (2007)


BindingDB Entry DOI: 10.7270/Q29Z9762
More data for this
Ligand-Target Pair