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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Lysine-specific demethylase 4C' and Ligand = 'BDBM347138'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Lysine-specific demethylase 4C


(Homo sapiens (Human))		BDBM347138
PNG
(2-(4-((2-methoxy-5-(4-methylpiperazin-1-yl) phenyl...)
Show SMILES COc1ccc(cc1N(C)c1ccc(Oc2nc(O)c3ccncc3n2)cc1C)N1CCN(C)CC1
Show InChI InChI=1S/C27H30N6O3/c1-18-15-20(36-27-29-22-17-28-10-9-21(22)26(34)30-27)6-7-23(18)32(3)24-16-19(5-8-25(24)35-4)33-13-11-31(2)12-14-33/h5-10,15-17H,11-14H2,1-4H3,(H,29,30,34)
PDB

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US Patent
n/an/a<100n/an/an/an/an/an/a



CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate-format under the following reaction conditions: 0.3 ...

US Patent US10202381 (2019)


BindingDB Entry DOI: 10.7270/Q2SX6GBM
More data for this
Ligand-Target Pair