Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Lysine-specific histone demethylase 1A (Homo sapiens (Human)) | BDBM50231780 (CHEMBL4065771) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 717 | n/a | n/a | n/a | n/a | n/a | n/a |
Key Laboratory of Technology of Drug Preparation (Zhengzhou University) Curated by ChEMBL | Assay Description Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assay | ACS Med Chem Lett 8: 384-389 (2017) Article DOI: 10.1021/acsmedchemlett.6b00423 BindingDB Entry DOI: 10.7270/Q2FQ9ZV3 | |||||||||||
More data for this Ligand-Target Pair |