Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Macrophage colony-stimulating factor 1 receptor' and Ligand = 'BDBM238229'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Macrophage colony-stimulating factor 1 receptor (Mus musculus (Mouse))	BDBM238229 (US9403804, 27) Show SMILES CC1(C)CCC(=CC1)c1cc(ccc1NC(=O)c1nc(c[nH]1)C#N)C1CCC(CC1)N1CCOCC1 |c:5,(5.16,7.26,;4.76,5.78,;6.25,5.38,;4.76,4.23,;3.43,3.47,;2.09,4.23,;2.09,5.78,;3.43,6.54,;.76,3.47,;.76,1.93,;-.58,1.15,;-1.91,1.93,;-1.91,3.47,;-.58,4.23,;-.58,5.78,;-1.91,6.54,;-1.91,8.08,;-3.24,5.78,;-3.24,4.23,;-4.72,3.72,;-5.61,5,;-4.71,6.25,;-5.2,2.26,;-5.67,.79,;-.58,-.38,;-1.91,-1.15,;-1.91,-2.69,;-.58,-3.47,;.76,-2.69,;.76,-1.15,;-.58,-5,;-1.91,-5.78,;-1.91,-7.31,;-.58,-8.08,;.76,-7.31,;.76,-5.78,)| Show InChI InChI=1S/C29H37N5O2/c1-29(2)11-9-21(10-12-29)25-17-22(20-3-6-24(7-4-20)34-13-15-36-16-14-34)5-8-26(25)33-28(35)27-31-19-23(18-30)32-27/h5,8-9,17,19-20,24H,3-4,6-7,10-16H2,1-2H3,(H,31,32)(H,33,35)	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.90	n/a	n/a	n/a	n/a	7.5	25
Janssen Pharmaceutica NV US Patent					Assay Description An autophosphorylation, fluorescence polarization competition immunoassay was used to determine the potency for c-fms inhibition exhibited by selecte...				US Patent US9403804 (2016) BindingDB Entry DOI: 10.7270/Q23T9G3C
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