Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Mast/stem cell growth factor receptor Kit [D816V]' and Ligand = 'BDBM392365'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Mast/stem cell growth factor receptor Kit [D816V] (Homo sapiens (Human))	BDBM392365 (5-fluoro-N-(2-phenyl-1H-pyrrolo [2,3-b]pyridin-5-y...) Show SMILES Fc1ccc2[nH]nc(C(=O)Nc3cnc4[nH]c(cc4c3)-c3ccccc3)c2c1 Show InChI InChI=1S/C21H14FN5O/c22-14-6-7-17-16(10-14)19(27-26-17)21(28)24-15-8-13-9-18(25-20(13)23-11-15)12-4-2-1-3-5-12/h1-11H,(H,23,25)(H,24,28)(H,26,27)	PDB UniProtKB/SwissProt GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	<1.00E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description Assays for biochemical cell-based activity of c-kit kinase are known in the art, for example, as described in U.S. Pat. Nos. 7,498,342 and 7,846,941,...				J Med Chem 52: 1799-802 (2009) BindingDB Entry DOI: 10.7270/Q2HH6NDZ
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