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Found 1 hit Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50106527'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM50106527
PNG
(CHEMBL3601031)
Show SMILES COc1ccc(cc1)-c1ccc(CCCNc2ccc(CN(C)C)cc2)nn1
Show InChI InChI=1S/C23H28N4O/c1-27(2)17-18-6-10-20(11-7-18)24-16-4-5-21-12-15-23(26-25-21)19-8-13-22(28-3)14-9-19/h6-15,24H,4-5,16-17H2,1-3H3
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n/an/a 154n/an/an/an/an/an/a



Boehringer Ingelheim Pharma GmbH& Co. KG

Curated by ChEMBL


Assay Description
Displacement of [125I-MCH] from human MCH receptor 1 expressed in CHO cell membranes by scintillation counting method

Bioorg Med Chem Lett 25: 3270-4 (2015)


Article DOI: 10.1016/j.bmcl.2015.05.074
BindingDB Entry DOI: 10.7270/Q2MK6FN7
More data for this
Ligand-Target Pair