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Found 1 hit Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50107757'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM50107757
PNG
(CHEMBL3601020)
Show SMILES Clc1ccc(cc1)-c1cnc(cn1)C#Cc1ccc(OCCN2CCCC2)cc1
Show InChI InChI=1S/C24H22ClN3O/c25-21-8-6-20(7-9-21)24-18-26-22(17-27-24)10-3-19-4-11-23(12-5-19)29-16-15-28-13-1-2-14-28/h4-9,11-12,17-18H,1-2,13-16H2
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Article
PubMed
n/an/a 17n/an/an/an/an/an/a



Boehringer Ingelheim Pharma GmbH& Co. KG

Curated by ChEMBL


Assay Description
Displacement of [125I]-MCH from human MCHR1 expressed in CHO/Galpha16 cell membranes by scintillation counting method

Bioorg Med Chem Lett 25: 3264-9 (2015)


Article DOI: 10.1016/j.bmcl.2015.05.077
BindingDB Entry DOI: 10.7270/Q25D8TMB
More data for this
Ligand-Target Pair