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Found 1 hit Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50107819'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM50107819
PNG
(CHEMBL3600390)
Show SMILES Clc1cccc(c1)-c1ccc(cc1)C(=O)NCCc1ccc(CN2CCCC2)cc1
Show InChI InChI=1S/C26H27ClN2O/c27-25-5-3-4-24(18-25)22-10-12-23(13-11-22)26(30)28-15-14-20-6-8-21(9-7-20)19-29-16-1-2-17-29/h3-13,18H,1-2,14-17,19H2,(H,28,30)
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Article
PubMed
n/an/a 29n/an/an/an/an/an/a



Boehringer Ingelheim Pharma GmbH& Co. KG

Curated by ChEMBL


Assay Description
Displacement of [125I]-MCH from human MCHR1 expressed in CHO/Galpha16 cell membranes by scintillation counting method

Bioorg Med Chem Lett 25: 3264-9 (2015)


Article DOI: 10.1016/j.bmcl.2015.05.077
BindingDB Entry DOI: 10.7270/Q25D8TMB
More data for this
Ligand-Target Pair