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Found 1 hit Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50107827'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM50107827
PNG
(CHEMBL3600824)
Show SMILES CCN(CC)CCOc1ccc(cc1)C#Cc1ccc(cn1)-c1ccc(OC)cc1
Show InChI InChI=1S/C26H28N2O2/c1-4-28(5-2)18-19-30-26-14-7-21(8-15-26)6-12-24-13-9-23(20-27-24)22-10-16-25(29-3)17-11-22/h7-11,13-17,20H,4-5,18-19H2,1-3H3
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Article
PubMed
n/an/a 35n/an/an/an/an/an/a



Boehringer Ingelheim Pharma GmbH& Co. KG

Curated by ChEMBL


Assay Description
Displacement of [125I]-MCH from human MCHR1 expressed in CHO/Galpha16 cell membranes by scintillation counting method

Bioorg Med Chem Lett 25: 3264-9 (2015)


Article DOI: 10.1016/j.bmcl.2015.05.077
BindingDB Entry DOI: 10.7270/Q25D8TMB
More data for this
Ligand-Target Pair