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Found 1 hit Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50153197'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM50153197
PNG
(CHEMBL184528 | N-(2-Diethylamino-ethyl)-4-[5-(4-ph...)
Show SMILES CCN(CC)CCNC(=O)c1ccc(cc1)-c1noc(n1)-c1ccc(Oc2ccccc2)cc1
Show InChI InChI=1S/C27H28N4O3/c1-3-31(4-2)19-18-28-26(32)21-12-10-20(11-13-21)25-29-27(34-30-25)22-14-16-24(17-15-22)33-23-8-6-5-7-9-23/h5-17H,3-4,18-19H2,1-2H3,(H,28,32)
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Article
PubMed
n/an/a 2.45E+3n/an/an/an/an/an/a



7TM Pharma A/S

Curated by ChEMBL


Assay Description
Binding affinity against human Melanin-concentrating hormone receptor 1 stably transfected CHO cells was determined using [125I]-MCH as radioligand

Bioorg Med Chem Lett 14: 5075-80 (2004)


Article DOI: 10.1016/j.bmcl.2004.07.077
BindingDB Entry DOI: 10.7270/Q2CF9PKT
More data for this
Ligand-Target Pair