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Found 1 hit Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50153216'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanin-concentrating hormone receptor 1


(Homo sapiens (Human))		BDBM50153216
PNG
(CHEMBL363264 | N-(1-Ethyl-pyrrolidin-2-ylmethyl)-4...)
Show SMILES CCN1CCCC1CNC(=O)c1ccc(cc1)-c1noc(n1)-c1ccc(Oc2ccccc2)cc1
Show InChI InChI=1S/C28H28N4O3/c1-2-32-18-6-7-23(32)19-29-27(33)21-12-10-20(11-13-21)26-30-28(35-31-26)22-14-16-25(17-15-22)34-24-8-4-3-5-9-24/h3-5,8-17,23H,2,6-7,18-19H2,1H3,(H,29,33)
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Article
PubMed
n/an/a 1.90E+3n/an/an/an/an/an/a



7TM Pharma A/S

Curated by ChEMBL


Assay Description
Binding affinity against human Melanin-concentrating hormone receptor 1 stably transfected CHO cells was determined using [125I]-MCH as radioligand

Bioorg Med Chem Lett 14: 5075-80 (2004)


Article DOI: 10.1016/j.bmcl.2004.07.077
BindingDB Entry DOI: 10.7270/Q2CF9PKT
More data for this
Ligand-Target Pair