Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Melanin-concentrating hormone receptor 2 (Homo sapiens (Human)) | BDBM50159343![]() (CHEMBL3787394) | Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >4.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Curated by ChEMBL | Assay Description Antagonist activity at human MCHR2 expressed in CHO cells after 60 to 75 mins by FLIPR assay | J Med Chem 59: 2497-511 (2016) Article DOI: 10.1021/acs.jmedchem.5b01654 BindingDB Entry DOI: 10.7270/Q23R0VSS | |||||||||||
More data for this Ligand-Target Pair |