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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM50202939'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Melanocortin receptor 4


(Homo sapiens (Human))		BDBM50202939
PNG
((+/-)-1-(2-biphenyl-2-ylethyl)-4-[2-(4-fluoropheny...)
Show SMILES CC(C)N1CCN(CC1)C(CN1CCN(CCc2ccccc2-c2ccccc2)CC1)c1ccc(F)cc1 |w:9.10|
Show InChI InChI=1S/C33H43FN4/c1-27(2)37-22-24-38(25-23-37)33(30-12-14-31(34)15-13-30)26-36-20-18-35(19-21-36)17-16-29-10-6-7-11-32(29)28-8-4-3-5-9-28/h3-15,27,33H,16-26H2,1-2H3
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Similars
Article
PubMed
n/an/a 186n/an/an/an/an/an/a



Taisho Pharmaceutical Co., Ltd

Curated by ChEMBL


Assay Description
Displacement of [125I]Nle4-D-Phe7-alpha-MSH from human MC4 receptor expressed in COS1 cells

Bioorg Med Chem 15: 1989-2005 (2007)


Article DOI: 10.1016/j.bmc.2006.12.039
BindingDB Entry DOI: 10.7270/Q2C53KHN
More data for this
Ligand-Target Pair